Introduction & Aims: Lower respiratory tract infections (LRTIs) are a leading cause of mortality worldwide [1]. Individuals with chronic respiratory diseases including cystic fibrosis (CF) are especially susceptible to LRTIs by bacterial pathogens such as Pseudomonas aeruginosa, which can become antimicrobial resistant (AMR) [2]. Bacteriophages (phages) are a promising alternative therapy against AMR infections; however, how phages retain their activity after delivery to the lungs via an aerosol is not well studied. For use as a therapeutic, <1 log10 reduction is considered a minimal loss of phage titre following aerosolisation [3, 4]. Here, we sought to test the effect of aerosolised delivery on the infectivity of P. aeruginosa phages.
Methods: Six phages (79.U1, 79.U2, 4.U3, E79, Boorn-mokiny-1, Kara-mokiny-16) from the Myoviridae family were individually nebulised using a vibrating-mesh nebuliser (Aerogen Pro). Nebulisation was performed into collection tubes to harvest aerosol condensate, infectious titre pre and post nebulisation was assessed via plaque assay of original and nebulised samples and expressed as plaque forming units per mL of sample (PFU/mL). Titre reduction values were compared to the acceptable level in the literature (<1 log10 reduction).
Results: Nebulisation resulted in a reduction of infectious titre for all six phages tested (values are presented as average log10 reduction ± SD PFU/mL) - KM-16: 0.49 ± 0.08, E79: 0.41 ± 0.13, BM-1: 0.11 ± 0.09, 4.U3: 0.27 ± 0.06, 79.U2: 0.20 ± 0.11, 79.U1: 0.08 ± 0.06. Loss of active phages ranged between 0.08 and 0.49 log10, below the acceptable threshold of loss for therapeutic use. In addition, reduction in infectivity for all nebulised phages was not significant (p > 0.05).
Conclusion: Phages can be aerosolised by vibrating-mesh nebulisation with minimal reduction in infectivity. Data generated suggests that aerosolisation is a feasible delivery method for phages against respiratory pathogens. Future work will test phages from various families to identify phage groups with high retention of activity in an aerosol, as well as buffers and adjuvants that may further stabilise phages during aerosolisation. Phage preparations will also be aerosolised with different delivery devices to ensure phage stability across a range of devices used by patients.